Pharmacology and The mechanism of action of Anastrozole

Pharmacological group: anti-estrogen drugs; non-steroidal aromatase inhibitors. Mode of action: the treatment of advanced breast cancer in women. Systematic (IUPAC) name: 2,2′- [5- (1H-1,2,4-triazol-1-ylmethyl) -1,3-phenylene] bis (2-methylpropanenitrile) Bioavailability: 83-85% Protein binding: 40% Metabolism 85% in the liver The half-life: 46.8 hours Isolation: 11% of renal Formula: C17H19N5 Mol. weight: 293.366 g / mol Anastrozole, available […]

Anastrozole in bodybuilding – courses and reviews

The main advantages Rapid suppression of aromatization The powerful inhibitory effect Inhibition of 50% of estrogen Increased levels of testosterone The lack of estrogenic activity Lack progestogenic activity High Absorption Non-steroidal drug Description Anastrozole – tableted preparation of the third generation, a potent inhibitor of aromatase. This highly selective non-steroidal drug is used in the […]