Pharmacology and The mechanism of action of Anastrozole

Pharmacological group: anti-estrogen drugs; non-steroidal aromatase inhibitors. Mode of action: the treatment of advanced breast cancer in women. Systematic (IUPAC) name: 2,2′- [5- (1H-1,2,4-triazol-1-ylmethyl) -1,3-phenylene] bis (2-methylpropanenitrile) Bioavailability: 83-85% Protein binding: 40% Metabolism 85% in the liver The half-life: 46.8 hours Isolation: 11% of renal Formula: C17H19N5 Mol. weight: 293.366 g / mol Anastrozole, available […]

Anastrozole: the use and side effects

Anastrozole (Anastrozole) – a powerful non-steroidal drugs used to suppress the phenomenon of depreciation. Anastrozole description. He acts, stopping the depreciation, as well as, ostanvlivaet body’s production of estrogen. Actually, he essentially differs from tamoxifen. It is only estrogen suppresses but does not prevent its occurrence. Anastrozole One dose Anastrozol lowers the amount of estradiol […]

Anastrozole or Letrozole: effective post-cycle therapy

The content of the article:   Action Anastrozole Application Side effects Anastrozole Women Letrozole in bodybuilding How to take Letrozole Letrozole for women   Among the athletes are very popular drugs such as aromatase inhibitors. These materials can improve anabolic hormones in the blood, to achieve relief, prevent hypertension. Meet with the best representatives of […]

Anastrozole in bodybuilding – courses and reviews

The main advantages Rapid suppression of aromatization The powerful inhibitory effect Inhibition of 50% of estrogen Increased levels of testosterone The lack of estrogenic activity Lack progestogenic activity High Absorption Non-steroidal drug Description Anastrozole – tableted preparation of the third generation, a potent inhibitor of aromatase. This highly selective non-steroidal drug is used in the […]

Anastrozole – comments on the application of the course in bodybuilding

Anastrozole – the new anti-estrogen agent, presented in oral form, based on the active ingredient Anastrozole. On the pharmacological market, it first appeared in 1995. Initially, anastrozole was used only for medical purposes: they conduct therapy of malignant mammary tumors with a high content of estrogen receptors. Now the tool in medicine is not widely […]

A brief description of Anastrozole

Anti estrogen drugs of the new generation. The main component – the active ingredient Anastrozole. For the first time the drug appeared on the market in 1995. First means are used exclusively for medical purposes. Anastrozole is used in the treatment of various tumors. Today in medicine drug is not widely applied. Basically anastrozololom are […]